99% Tianeptine sodium munyu CAS 30123-17-2
Tsanangudzo
ITEM | STANDARD | RESULT |
Chitarisiko | Hupfu hwakachena kusvika kune yero | White crystalline powder |
Solubility | Freetly soluble Mumvura uye methanol uye dichloromethane | Conforms |
Identification | Ne IR, Kuenderana neyakajairwa kushanda | Conforms |
(2) Inopa maitiro e sodium | Conforms | |
Zvisina kuchena A | ≤0.1% | Haisati yaonekwa |
Related compounds | Chero Max kusachena kumwe chete≤0.1% | 0.060% |
Zvose zvisina kuchena≤0.4% | 0.36% | |
Residual Solvents (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Methanol≤ 0.3% | ND | |
Acetone≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Mvura | ≤ 5.0% | 3.8% |
Kuongorora (HPLC) | 99.0% -101.0% (Paanhydrousbasis) | 99.70% |
Application
Tianeptine sodiummunyuinonzi tricyclic antidepressant.Maitiro ayo ekurwisa kushushikana kwakasiyana neaya echinyakare tricyclic antidepressants.Inogona kuwedzera kudzokororwa kwe5-HT mune synaptic cleft.Migumisiro yeHT neuronal conduction.Hapana hukama hwecholine kana adrenergic receptors.Iyo antidepressant efficacy yakafanana neye tricyclics, asi kushivirira kuri nani pane iyo ye tricyclics.Kurapa kwekuora mwoyo kwakapfava, kwakadzikama kana kwakanyanya, neurogenic uye reactive depression, kuzvidya mwoyo uye kuora mwoyo nemuviri, kunyanya kusagadzikana kwepamuviri, uye kushungurudzika uye kuora mwoyo muvarwere vanodhakwa panguva yekurega.